Ola kinoHoomakaukau

"Montelukast": hōʻike manaʻo, olelo ao a me analogues o ka lāʻau

"Montelukast" - e pili ana i ka lāʻau 'hōʻike manaʻo hiki wale ke loaʻa i online, Usenet a me nā mea laʻa a kahua i ka pilikia o ka asthma - he Classic hoa o ka leukotriene D4-mea loaʻa. Ka lāʻau 'Ua hoʻomano hoʻohana me ke kumu ma ka Inc, a i ole ano ino o ka maʻi. Balanced haku mele 'apono' i ka hoʻohana 'ana i ka lāʻau no ka iapaau ana o nā mea maʻi o ka aneane kekahi makahiki pae.

hookuu palapala

Kumu "montelukast" loaa ka hapanui oluʻolu nāʻana, he hailona. Naʻe, i ka mea mua e catches kou maka - keia mea, o ka papa, he assortment o na papa, a kuai lilo aku ma lalo o ka inoa kalepa o nā ikepili.

Ma ka manawa o ka kaʻina ua Kīwala'ō ma lalo ekolu'ōpū mai. Ua mea e pili ana i ka hae huaale me ka pepa kini wahī (1 pa alima he 10 mg oʻeleu waiwai) a me kā lākou mau analogues kamaiʻilio (4 mg a me 5 mg pakahi o ka mea kemikala). Base kumu i loko o nā hihia, hana montelukast paʻakai, akā, no ka haku mele 'ana o kekahi mau' ano 'okoʻa kākoʻo eiiiiiaiou - Mannitol a me aspartame i noho i loko o kekahi laʻana manao ia no ka' ai, inu koke i hoʻohana.

Ma muli o kona kulana manaʻo pinepine ia POP i ka ninau o counterfeits, i kēia manawa, a laila,ʻikeʻia ma ka hale kūʻai lāʻau lapaʻau na kaulahao. Hoku Welowelo ku counterfeiting hiki ia, ina e 'eleu uku hoʻolohe i ke ano o ka pharmacological huahana.

Ma kekahi, e kamaiʻilio ana Akala a me 4 milligrams oʻeleu 'Oponopono, mai ka'ololaha shape a me ka tinge nonono (hōʻikeʻano hoʻopili like papa me ka kamako ikiʻono, a me ka hoʻohana' ana i nā flavorings ana oko ao), a ia ia me ka nui "4" ma kekahiʻaoʻao. Analogs ma i ka papa kuhikuhiEʻeleu 'Oponopono mea 1 mg hou - a me ka' ae ' "elima". Akala like me ka iwi geometrically e hoohalike ai i ka rectangle; Ka mea, beige a helu "10" helu.

pharmacological affiliation

"Montelukast" (kūmole hōʻike no wahi, i hiki i kahi luna 'mea kemikala hoʻonāukiuki allergies i loa pohihihi) - keia mea he typical ka Luna o ka pae antibronhokonstriktornyh ai'. Ke algorithm e leie aku kona hana, e olelo aku i ka "kokoke pilina" me ka intermedianty / prostaglandins a me thromboxanes.

O ka papa kuhikuhi hana o ka lāʻau - ka paleʻana cysteinyl leukotriene "nā mea e loaʻa ka mea nalo" o ka naehana nenoaiu. Mau receptors mālama kiʻekiʻe haʻawina i loko o bronchial asthma ulu a me ka mea hoʻoulu i ka hoʻololi kemikala o secretions a laila accumulates a complicates ka mucosa.

Ka pololei,ʻai anaʻo ia i ka nui ka ho'ēmiʻana i loko o ka oolea o symptoms ma ke kāʻei kua o ka mau emi ana i loko o ka helu o ka asthma ho'āhewa wale (i kaulana e na mea he nui nā mea maʻi, maikaʻi nā loli i ua ike i ka lā mua o ka Inc).

metabolic hiʻona

"Montelukast" (hōʻike manaʻo pharmacists paipai i ka maoli i waeia o ka oukou e ku-ins mea i kaupalena 'ia ke kumu kuai pilikino E pili ana i Manufacturers, oa ke kanaka ai'-synonyms, Ua haawiia i kona haku mele 'ana'ālike-mea kūkulu nā lātoma i ka papa kuhikuhiE ke keʻena, ma laila i kekahi mau manawa oi pipiʻi ma mua o ka mea i ho'ākāka' ia e hoomakaukau ai), komo i loko o ka wai koko ke koko, e hoopaa ana hoʻi mai kēlā wahi a me kona nā polokina. Ma lapaʻau haʻawina, i kākau i ka hopena i 99, 37%. I ka Ia manawa, kona bioavailability mea ma ka pololei e like me ke kaʻina hana o ka issuance. No ka laʻana, na nā mea hoʻohui 5-milligram papa amenable ke omo ma ka 73%, no ka mea hoi analogues me kaʻili lahilahi liner ma a he mea 2 manawa houʻeleu waiwai, - wale ma ka 64%.

A like kulana home 'ole me ka hapa-ola o ka mea kemikala: eiiiiiaiou e kamaiʻilio ana huaale, ma ka undergoing pūnao, e waiho ana i ke kino ma hope o 2 hora hope? Eaia, akā, i ka constituent kumu o kaʻike mau papa - ma hope o 180-200 minuke. Ma keia wai kokoʻae loli aʻe ma waena o 43-45 ml / minuke. A, interestingly, wale 0.2% o ka mahele lāʻau ua haliiaʻe urinary kaha. Naʻau liʻiliʻi, ma ka nane hea, - oi ma mua o 85%.

Mai ka loa o ka hanohano Aupuni, ka mea, penei i ka pharmacokinetic kaʻina mea like smoothly i loko o nā mea maʻi o nā sexes, a me ka mea e kekahi mau hoʻoponopono 'kaumaha no ka makahiki a me kaʻaʻa puʻuwai pathology ma ka i ka ho omaulia ana o ka mea i kela la e lawelawe ana o ka lapaʻauʻia ua koi' ia. Akā, me ka ole o ke akepaa, o ka oi aku ka wā e hele i ka loa mai, hewaʻiʻo nānā 'ana i ka makaukau ana o ka pākōlea haʻalele' ana.

nāʻikepili no ka

I ka hoaponoia ma ka hoʻohana 'ana o "montelukast" lāʻau hōʻike manaʻo (keiki ka lapaʻauʻia e waiho i loko o ka palapala o ka nui aʻe ana, huaale, kapa komo iā iaʻili lahilahi iwi, ia mea kupono e hoonoho wale nō nā mākua a me nā adolescents), haʻalele ma Usenet, o ka papa, kōkua iā mākou e maopopo. Eia naʻe, wale alakaʻi ma ka manao nā poʻe o - ia mea he nui kuhihewa, no ka mea, me ke kūkā pū me ka kahuna lapaau, "e hōʻike i ka" 'ano o ka asthma, a me ka hapanui importantly - e loaʻa mai i ke kumu no kona hanana mea aneane hiki ole i.

Me ka pili ana i ka oihana hoakaka, ka p ÷ ai ma laila symptoms, maʻi puʻuwai a me nā kūlana o ua hōʻolokeʻaʻia like penei:

  • bronchial spasms triggered e excessive physical haawe;
  • Naciiiuo / maʻi rhinitis, allergic ano o ke kumu;
  • asthma;
  • i ka pono no ka kāohi ana.

Na kaʻoi loa laʻau heluna

"Montelukast" (io manaʻo mea paʻakikī loa e loaʻa, no ka mea, o kaʻeleu 'Oponopono ua lōʻihi ua ana hoʻohana like me ka' ōlelo ke keʻena o ka nui lāʻau) ua lawelawe hōʻike waha, hookahi manawa i ka lā, me ka hana ana i ka haʻalele 'ana "aina kakahiaka - aina awakea -. Awakea"

No ka chewable na papa, 4 mg a me 5 mg ka poe hana pela dosages rula:

  • keiki kahiko ma waena o 2 a me 5 makahiki: 1 pa alima o ka huahana (4 mg) i ka lā, ma bedtime, a loaʻa hooponopono ana o symptoms a me prolongation o ka muli o papa no 2-4 pule, e koho i ka resultant hopena;
  • hoʻomanawanui iki mai 6 i ka 14 o kona mau makahiki:ʻo ia pololei, akā, he hoʻokahi-manawa uku o - 5 mg.

No ka huaale me ka pepa kini wrapper pili i kēia koi:

  • mākua a me nā keiki ma luna o ka 15 o kona mau makahiki, e loaa ana mai ka bronchial asthma a maʻi rhinitis: 1 Unit (10 mg o ka mea) / lā i loko o ke ahiahi;
  • e pale aku cramps:ʻo ia mahele lāʻau ma luna o kekahi manawa wā mawaena lōʻihi o 14-28 lā.

ʻaoʻao kanawai

"Montelukast" aʻo (hōʻike manaʻo paipai i ke ahiahi, i piha kaʻaeʻana me nā kūhelu alakaʻi o atypical reactions a hiki i ke alo o nā mea hoʻohui a hiki i ka hopena,ʻaʻole hiki ke ā) ua hoʻonoho like me ka palena papaha palekana lāʻau, akā, me ka proviso i ka ole-i ho'ākāka ' "muli o" ma ka aoao o ke kino i loko o kēia hihia nō e hiki.

Aeia mai ha:

  • GI: diarrhea, maloo waha,ʻeha ma ka abdomen maʻi pale, nausea;
  • naau a me ke koko laina: he loa nui mahuahua ma ka lāʻau ikiʻai wale kōmi;
  • ili poʻe noʻonoʻoʻole, urticaria, kūloko hematoma;
  • naehana'ōnaehana: runny ihu, a me ka puʻu;
  • CNS: pōniuniu, luhi, naʻau i loko o ke kaumaha alternating me excessive psychomotor manaʻo pīhoihoi;
  • musculoskeletal: myalgia a me ka arthralgia (me convulsions.).
  • Other: symptoms ano o ka huʻi naehana nā mea palahēhē a me ka maʻi palū.

Hoʻokau 'a me contraindications

"Montelukast" (kuhi no ka pomaikai o ka loa 'oluʻolu hōʻike manaʻo, a me ka ike iloko o loko o laila, ma ka hua'ōlelo o ka objectivity, ninau mai lālā o ka waihona mea kokoke,ʻaʻole ma laila),ʻaʻole e pili inā:

  • Ua loaʻa he mahuahua pā lonoaʻili i ka haku mele 'ana o ka laau (ano laulā, oiaio no a pau ano o ka papa);
  • diagnosed pohihihi keia ili maʻi, a me ka poʻe i loko o a ka meaola aʻole i assimilate galactose aʻike piʻi noho pilikia lactase deficiency (keia kapu, aole ia e pili i ka kamaiʻilio huaale);
  • ka hoʻomanawanui ua kaumaha me phenylketonuria;
  • ka hoʻomanawanui i ole i huli elua makahiki (no ka lole komoʻuʻuku nona na papa io "makahiki kali" - 15 makahiki).

Overdose: Symptoms a me ka lapaʻau

Hawaiʻi Ua hōʻike, "Montelukast" 4 mg (i maopopo nä haumäna e pili ana i keia kalepa palapala o ka mea kemikala, ma ka mea,'ālike i nā manaʻo i mea e kamaʻilio aku e kamaiʻilio ana analogs i loaʻa ka 5 mg oʻeleu waiwai) ma ka oi o ka i kela la hokii uku i ma luna o ka mea ia ia me 10 mg papa . Ka loa haʻi symptoms o overdose hiki ke ike i loko o nā mea maʻi kaikaina pae. Mākua, i ka wā e lawe 200 mg / lā no 5 mahina, i mālama kekahi'āno'ē reactions.

Ka hookahi hoailona Episode o ka mahuahua nā hoʻohui like o ka lāʻau i:

  • pio ole o ka make wai;
  • drowsiness;
  • opu wahi eha;
  • ka luaʻi;

Lapaʻau ua lawe mai, ma muli o ka lapaʻau kiʻi malama. Information e pili ana i ka laulā o ka hemodialysis kahi e.

Uluwehi O hana kūleʻa, a me ka loa Popular analogues

"Montelukast" 5 mg (hōʻike manaʻo o kamaiʻilio Eia kekahi laʻana haʻalele ma pediatricians, hoʻolapalapa i lalo i ka manaʻo i ka lāʻau, i lana ai, e pono no i ka noonoo ana o na makua opiopio), e like me nā ano o ka leukotriene mea loaʻa hoa, ka wā hoʻohana i ia laua me ka pili Luna e hōʻeleu i ka maikaʻiʻano : symptoms o asthma i emi loa, i ka helu o ka ho'āhewa wale ua hoʻemi. Naʻe, i ka abrupt withdrawal o Inc lawe mai ma luna o ka muli o ana corticosteroids ua ole paipai.

Nui likeʻole i loko o ka pharmacokinetic keʻano o ka hanaʻana pili i theophylline a me ka prednizola akomi i. Akā, omo i "hoao ana" me ka phenobarbital emi ma ka like ka nui me 40%.

Reagents i inhibit ka hoʻololi kemikala o CYP3A4 isoenzyme, E e hoʻohana ma lalo o 'inikua hooponopono wale.

Mall analogs i ka loa pinepine loaʻa ma luna o kuai:

  • "Monkasta".
  • "Singlon".
  • "Singulair".
  • "Ektalust".
  • "Singuleks".

"Singulair" a me "montelukast": hōʻike manaʻo o nā kauka, a pharmacists

E like me ke akamai pharmacologists, hoopaapaa e pili ana i o ka ai 'ka lua pele a me ka oi ka hoʻokō, meaningless, no ka "Singulair" a me ka "montelukast" i kekahi a me na ia mea lāʻau lapaʻau kumu. Iki hala ka mua kalepa inoa iaoaioa helu, a me ka lua o ka mea lahui. Kanaka kahuna lapaau a me nā mea maʻi, eia nae, i ka okoa e nānā, a noonoo ka lapaʻauʻia haawi ma lalo o ka hale kipa, ka mea wale pololei olelo hooholo.

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