Ola kinoHoomakaukau

"Relpaks": aʻo no ka hoʻohana, nāʻana. lāʻau analogues

Migraines, aole nae i ke ola hooweliweli kanaka e loaa ana ia, akā, i ka mea ia manawa me ka nui loa ho'ēmi i kā ka mea e like ai o ke ola. Over o ka makahiki, i nā mea lāʻau lapaʻau ka hana e hana ana i ka ho okumu ana i nā huahana i makemake ole hoʻopau wale i ka eha symptoms o kēia maʻi, akā, no hoi, e ho ololi i ka keʻano o ka hanaʻana i i ka migraine. Ma hope o nā mea a pau, e hooki i kaʻeha hiki e ikaika painkillers. Akā, 'ē aʻe symptoms o migraine e like me nausea, malamalama pā lonoaʻili a me ka intolerance i ka mea kani-, ia mea i oluolu i ka hoʻopau. Ka lāʻau no ka migraine "Relpaks" ma keia manao, poe akamai i olelo aku kekahi o ka loa ka hoʻokō. He aha ka keia k? Pehea e lawe ia, a mea i kona counterparts ma laila? A pau i kēia 'oe ke heluhelu ma lalo nei.

hoʻomanaʻo hōʻikeʻano

I ka papa kuhikuhiEʻeleu waiwai "Relpaks" e hoomakaukau ai - i loko o ka palapala o ka eletriptan hydrobromide ua hookomoia ma ka papa o ka 20 mg. Aia mea no hoi kekahi laʻau heluna o 40 mg. Auxiliaries i olelo ia i loko o ka mea lāʻau lapaʻau hana lactose monohydrate, makanekiuma stearate, croscarmellose paʻakai a me MCC. Mau i huiʻia mai,ʻaʻole pili i ka hiki ana o ka lāʻau a hiki i ka digestion, a aole i pili i ke kino e like me ke okoa. O na papa io o ka migraine "Relpaks" kapa komo iā iaʻili lahilahi iwi alani, a he titanium'okikene lua, colorants, lactose monohydrate, hypromellose a me ka triacetin.

Kēlā me kēia papa ua hanaʻia i loko o ka poepoe biconvex shape. Ma kekahiʻaoʻao ka mea, ua kii o «Rep 20» a «Rep 40 '(ke kaumaha ma muli o ka nui i loko o ka papa o kaʻeleu' Oponopono) a« Pfizer »- i kekahi. I kekahi blister fits 2, 3, 4, 6 a 10 na papa, a, ma ka huli, piha ma ka pepa pahu 1, 2, 3, 4, 5, 6 a 10 apana.

Pharmacokinetics a me pharmacodynamics

koke, a pono ke kemu Medicine "Relpaks" ma hope o ku una hooponopono, pakahi aku la ia i loko o ka hui pu ana me ka momoma ka ai. Omo eletriptan averages ma kahi o 81%, a me ka ai-kapaia bioavailability - 50%. ʻO kā mākou maʻiʻo o kaʻeleu waiwai i loko o ke koko wai koko mea mua kekahi, a me ka hapalua hola e lawe i ka lāʻau ma hope.

I ka papa kuhikuhiEʻeleu waiwai "Relpaks" e hoomakaukau ai i ka hana ana i ka pono no ka pili ana me ka wai koko nā polokina (ma kahi o 85%). N eletriptan pūnao ia lŘlŘ ma ke akepaʻa keena. Pela i hana mau ai hoʻolahaʻia metabolite, hoʻokahi (i hanaʻia e N-'okesaside)ʻaʻohe ha awina. Ka lua (i hanaʻia i loko o ka N-demethylation) i kekahi o ia waiwai, e like me ka palapalaʻia, akā, kona lehulehu ma ka wai koko mea wale 10-20% o ka lehulehu o ka eletriptan. Aie i kaʻeleu metabolite aole appreciable pākōlea hopena.

Papa migraine "Relpaks" pane o ka poe akamai i i i ka hapanui 'oluʻolu, ka hoʻokō nānā' ole o ka wahine o ka hoʻomanawanui. Excretion o ka lāʻau metabolites ua hana mai ia i ka nui loa ma nā puʻupaʻa (ka hola 90%), a ma ka naʻau liʻiliʻi.

Haʻawina i hoopaa i ka nele o ka hookoia ana o habituation i ka papa kuhikuhiEʻeleu 'Oponopono o ka lāʻau, no laila, ua loaʻa heʻaʻohe kapu ma luna o ka lōʻihi like' ole o ka Inc o migraine eha ma ka hoʻohana 'ana i ai' "Relpaks".

KŘpa a pharmacodynamic lāʻau "Relpaks" hoʻohana noi Shoes i ka mea i kona papa kuhikuhiEʻeleu waiwai no a hiki i ka pae ana e wae serotonin vascular a me neuronal receptors, ka lawe 'ole ma nā' ano o ia mau mea. Pela selectivity ua hoikea mai oia, a hiki i ka nui loa pili i na receptors aia i loko o ka carotid arteries. Protivomengrinoznuyu ha awina eletriptan hoʻoholo ole wale kona hiki i ka hou ana o ka moku koko aia i loko o ka cranium, akā, i ka maikaʻi ia ma luna o ke ano o neurogenic li nui. Ma keia hihia, me kaʻeleu waiwai i kokoke ole ia ma luna o nā receptors o ka femoral a me ka coronary arteries.

hoike

Uluwehi O "Relpaks" kauoha no ka hoʻohana 'e waiho ana ma na ano mau o ka migraine:

  1. Me ka aura ka wā i hoʻohuiʻia ai i ka loaʻeha symptoms e like me pilikia makapō, tactile, Hawaii, olfactory a me auditory kāna hana.
  2. Me ka aura, ka wā i hou i ka headache ahonui e pili ana nausea, ka luaʻi, pā lonoaʻili i ka malamalama a me ke kani.

Inā he mea 'ē aʻe ano o ka maʻi i ka hoʻohana' ana i ka lāʻau,ʻaʻole wale mai i ka maikaʻi ia, akā, hiki no hoi i kekahi mau complications. No laila, ma mua oe e hoʻohana i kēia lāʻau, e hoʻopau i ka headache, migraine, e pono e nīnau i ka hoʻomalu, a undergo piha ninaninau. Kēia e kōkua ole wale no i hoakaka ia e pono lapaʻau, akā, no hoi, e hoʻopau i kamepiula koke i ke ola o ka hoʻomanawanui.

Contraindications

E noonoo i ka papa inoa o nā contraindications no i "Relpaks" lāʻau. Na papa, e like me ka olelo maluna, no eletriptan i mea hiki ke systemic 'ole ma o ka meaola a ololi he nui keʻano o ka hanaʻana. Ma kekahi mau hihia, ka hoʻohana 'ana i ka huina hoonui unacceptable paha undesirable:

  • ma ke alo o ka kiʻekiʻe e pā lonoaʻili o ka hoʻomanawanui i nā mea a pau 'ona ho okumu i kekahi hapa o ka lāʻau;
  • i loko o kāna hana o ke ake, a konāhua, me pūnao a me excretion o ka papa hana 'Oponopono ia lŘlŘ i loko o ia mau mea;
  • me ka kipi hypertension;
  • me ka latent paha Puhi iho awa maʻi o ka naau, me ka naau hoouka, angina, coronary artery maʻi;
  • ma ke alo inklyuzionnyhʻike ākea vascular maʻi;
  • ka wā hoolilo paha na ma ka manawa o ka transient ischemic kaua, e like me kekahi 'aʻe' ana o cerebral holo.

Uluwehi O "Relpaks" categorically i paipai no ke kanaka nona ka makahiki ka emi o na makahiki 18. Eia kekahi, i ka lāʻau 'hiki ole ke ia no ka kokua o kaʻeha hou pili i ka headaches na migraineʻano like basilar, ophthalmic a me ka hemiplegic.

E hoʻohana i hāpai keiki, a lactation

E ho ohana ana o ka lāʻau "Relpaks" i hāpai keiki i ua insufficiently? Anoee. Eia naʻe, keʻena hoʻokolohua haʻawina ma holoholona hōʻike i ka hopena o ka eletriptan ma luna o ka ulu fetus. Mua, ua 'akomi i ka uuku o mutated nā'ōewe (e like me ka rula o ka polyploidy) i loko o ka embryo. ʻO ka lua, he piha-manawa hanau ke kaupaonaʻana ua me ka nui loa haʻahaʻa ma mua o ka holoholona i i ole loaa i gestation eletriptan. A no ke aha la akamai i loko o kona manawa i oleloia ai alakaʻi rula, i mea e ka pōmaikaʻi kakali ana i ai i ka makuahine, ma mua o ka hiki wā e hiki mai ka pilikia a hiki i ka fetus. It E e kaulana ia eletriptan, hapa o ka lāʻau i loaʻa i loko o kanaka ka waiū, a hiki ma hope lā ma hope? Eaia. No laila, i ka hoʻohana 'ia o ka lapaʻauʻia ma ka poe makuwahine mea hiki wale i ka hihia o ka hoʻokō' ole 'e breastfeed no ma ka liʻiliʻi loa o ka lā.

ʻaoʻao waiwai pili me ka lāʻau i "Relpaks"

Portability "Relpaks" lāʻau hōʻike manaʻo hoʻomalu i ka 'ike e pili ana i nawaliwali ka oolea o kaʻaoʻao waiwai, i wale nō i loko o ka kŘpa a pōkole wā o ka manawa. Ia, aole i nui ka mahele lāʻau (20 mg 'ole 40) i loaa mai ma o ka hoʻomanawanui. Ka loa, he pono ole symptoms ua hoano e ia e lawe i ka lāʻau e:

  • li nui o ka nasal lua a me ka pharynx (pharyngitis, a me ka rhinitis);
  • sensory haunaele e like me tingling, "Oie bumps";
  • drowsiness;
  • pōniuniu paha headache;
  • myasthenia gravis ole hypoesthesia;
  • hypertonicity o ka Muscle olona,;
  • ka eha, a me ka manao pono i ka hope a me ka umauma;
  • cardiac arrhythmias, i loko o ua tachycardia;
  • dyspeptic kāna hana e like me ka eha a discomfort i loko o ka abdomen, maloo waha , a me ka nausea;
  • mahuahua ma ka sweating;
  • wela flushes ai ole, e he maka.

Lālau aʻela ia i loko o ka mooolelo o ka Nine Inch haku mele 'o "Relpaks", mākaukau mai i hookaawale ia i ka hooulu ana o allergic reactions i eiiiiiaiou o ka lāʻau, a hiki e hoikeia ma ke ano o ka poʻe noʻonoʻoʻole, maneo a redness. Eia hou kekahi, ma ka pohihihi keia hoopii, nā mea maʻi i e hopohopo e pili ana i kaʻike manaʻo like:

  • anorexia;
  • lymphadenopathy;
  • ka hilahila, euphoria a kaumaha, Kanikani'āʻula. a me ka 'ehaʻeha o lability;
  • photophobia,ʻeha i loko o ka'ōnohi a poʻopoʻo, conjunctivitis, hoemiia paha mahuahua lacrimation;
  • hoao dysfunction;
  • ringing i loko o nā pepeiao, a soreness;
  • kiʻekiʻe ke koko;
  • asthma ho'āhewa wale;
  • hoʻololi i ka leo leo;
  • haanou ana i ka moʻolelo o ka lua;
  • constipation paha diarrhea;
  • arthritis paha arthrosis;
  • myalgia paha myopathy;
  • polyuria a pinepine urination;
  • menstrual kāna hana;
  • ischemic colitis.

Lālau aʻela ia i loko o ka mooolelo o ka luna-i oleloiaʻaoʻao 'ole, ka hoʻohana' ana o kekahiʻano o ka migraine "Relpaks" Ua pono, e lawe mai ma lalo o ka hooponopono ana o poe akamai, a me ka wale ma hope o ka mea e pono haʻawina no na maʻi e e lawe mai, a hiki complicate lapaau.

AaOIeIOUIeXAOAaIN

E noonoo oe i ka AaOIeIOUIeXAOAaIN me kekahi ai 'antimigraine konohiki "Relpaks". Ka lapaʻauʻia alakaʻi a he nui 'ike e pili ana i kona hoʻokaulike me nā ai' e ole e lawe pu ia me ka mea e pono ai ka lapaʻauʻia kēia mau pūʻulu.

  • isozyme nā mea kūpale, a loaʻa "erythromycin", "ketoconazole" "Clarithromycin" a me ka "Itraconazole";
  • protease nā mea kūpale, a me "nelfinavir" a me ka "Indinavir".

Akamai no hoi e hoailona oukou i ka mea i ka i ka wā hoʻokahi? Eaia "Relpaks" lāʻau lapaau "Propanolol" a me ka "Verapamil" hiki hoonaukiuki wale ka nui mahuahua i loko o ke koko,, akā, i ka hōʻoi 'i ka pilikia o nāʻaoʻao loa. Hoʻonuiʻia ke koko, hiki ke manaoia ma ka hihia o ami pono o ka lāʻau me ka caffeine ai '. A no ke aha la poe akamai i waiho aku i kela la i keia wā mawaena ma waena o? Eaia o na ai 'like "Relpaks" (i haule analogues ma lalo o kēia ho'ākāka' ana) i a me ka ergotaminopodobnyh ai '.

Clinically, ka mea, ua hoao aku au ia i na mea o ka migraine ma ka ninau i loko o keia 'atikala' Aʻole i pane koke me ka waiwai e pili ana i ka Hoʻokolohua-blockers, estrogensoderjath hōmona hope paha waha contraceptives, akā, no hoi a hiki i ka tricyclic antidepressants.

overdose

Inā 'oe mamua o ka paipai kauka dala o ka lāʻau "Relpaks" manual ao o ka overdose, a hiki i ka pinepine mahuahua ana i loko o ke koko, a me ka' ē aʻe kāna hana o ka mea'ōnaehana mānowai koko nenoaiu. A hiki aku ka mea, hōʻike a me ka symptomatic hana ua paipai ina e pono ai gastric lavage.

Dosing

Uluwehi O "Relpaks" poe akamai i Paipai 'e lawe i ka hoʻomaka o ka migraine ho'āhewa wale. Inā ka headache a me nā maʻi puʻuwai conjugate ia bother i ke ahonui no kekahi mau hola, e like me ka lāʻau i hoopaa mai ai kona laulā. It E e kaulana i? Eaia o ka lāʻau 'like me ka kāohi Agena no ka migraine mea inexpedient, no ka mea, ua hoao aku au ia ia i loko o keia hihia ka mea,' aʻole i loaʻa ka mea i makemake ia. I ka Ia manawa, i ka wa e nee mai ana i ka aura (nā mea maʻi, lōʻihi-makahiki migraine sufferers ke kuhikuhi keia kulana) e lawe i ka lāʻau 'ole ho'ēmi i kā wale i ka eha ana ma hope o ka aura, akā, i relieves symptoms e like me nausea, drowsiness a me ka photosensitivity. i keia ia lŘlŘ kekahi manawa, akā, ma hope o ka hoouka kaua ana o headaches wale. Nolaila, migraine sufferers e ole mai oukou, mailoko e inu i ka Akala a kēlā me kēia manawa i ka maʻi puʻuwai.

I ka loiloi mua mahele lāʻau o ka lāʻau no nā mea maʻi 18-65 makahiki o ka makahiki, he 40 mg. Ma hope iho o ke kokua ana o migraineʻeha hiki ke laila. Ma keia hihia, ke alakai i ke heluhelu lawe i ka lāʻau hou ma ka ia laʻau heluna, akā,ʻaʻole koke ma mua o 2 hola ma hope o ka hiki mua. I Ina o ka hoʻokō 'ole' ana i ka lāʻau 'ka wā headache unabated iloko 2 hola ma hope o ka lāʻau hooponopono, hou-ana ua i paipai mahele lāʻau. Ke hoʻomalu kuhikuhi mai i ka mea e hiki mai ana hoouka o migraine i loko o ka ua hoʻomanawanui hiki ke docked loiloi mua mahele lāʻau "Relpaks" lāʻau. Consumer hōʻike manaʻo ma keia manawa no hoi aia no iloko olaila ano like 'ike.

ʻO kā mākou mahele lāʻau o ka medicament i loaa i loko o ka lā hoʻokahi e ole oi 160 mg. Inu papa e e ola, me ka e kamaiʻilio ana, inu nui o fluids.

Cautions

Ka hoʻohana o "Relpaks 'hoomalolo mea hiki ma hope o ka hōʻoiaʻiʻo nō o kaʻike, a wale" migraine ". O ke kumu ho i ka mea i ka wā atypical headaches, i hiki ke kena ae la no hoi ma ka hahauʻana, aneurysm rupture a me nā maʻi nui, kona hookohu ia ke kāhea likeʻole complications. Eia kekahi, ia mea undesirable e hoʻohana 'ia k ‰ e hoʻopau loa kaʻeha ma ka migraine amid mea'ōnaehana mānowai koko maʻi a me kāna hana o ka hakuʻala a me akepaa, me keia hiki i kiʻekiʻe ke koko, a hiki i ka pilikia kiʻekiʻe. ʻO ia pili i nā mea maʻi i loko o ka mea a ka pilikia o ka ulu mea'ōnaehana mānowai koko maʻi mea kiʻekiʻe. Ia mea ke kumu mua e ho'ākākaʻia ka lāʻau "Relpaks" ka hoʻomanawanui E undergo i ka piha ninaninau. Nā mea maʻi i hoʻohana no 65 makahiki o ka lāʻau e ia ma lalo o ka hooponopono ana o poe akamai, no ka mea, o ka mea, loa pinepine ia malama mahuahua i loko o ke koko,.

Aʻo! E pili ana i ka? Eaia o ka lāʻau "Relpaks" manual kekahi i maopopo nä haumäna i kaʻaoʻao 'ole me pōniuniu a me ka drowsiness, pela no oe e e oi loa akahele kaa ka wā e hoohauhee ana a me ka mālama' ana i ka 'enehana luna'.

Analogs "Relpaks" lāʻau kumukuai

I ka hapanui o ka ai 'i lawe ma ka mea lāʻau lapaʻau poʻe i loko o ka West, he mau wahi lulu counterparts. Mākou ke'ōlelo e pili ana, a ku e Pfizer - ka hoʻohua "Relpaks" lāʻau. Eia naʻe, no ka mea, ua kakau wale nei, i ka lā ma laila nō ole ai 'i makemake i ka ia waiwai e like me ka lāʻau "Relpaks". Analogs ka papa kuhikuhiEʻeleu 'Oponopono eletriptan iʻikeʻia, mai i ka mea hiki ke manao ia o ka la hoomalolo mea kū hoʻokahi. kona kāki ma Rusia mea mai ka 380 a hiki i 1200 rubles. Ka mea i ho'ākāka 'kumukuai hilinaʻi nui ma luna o ka helu ana o na papa i loko o ka AEeAaOA a me ka mea kā lākou laʻau heluna.

Ma ke ano o ka hopena ma luna o nā ipu lolo ma ka papa "Relpaks" loaʻa nō kekahi mau counterparts, i ole wale mai oko nui mai ia ia i waiwai e lilo aku, akā, ua ikaika nui ae pipiʻi pinepine. No ka laʻana, o ka laau no ka migraine "Zomig" hiki ke kuai ma kekahi kumu kuai o ka puni 400 rubles no ekolu huaale. Ai ' "Imigran" a me ka "Sumatriptan" mea i like loa ke "Relpaksom" i ke kanawai o ke a me ka uku. Ke wale lāʻau, i loaʻa nui i emi ma mua o "Relpaks" papa - he "Kofetamin". Lākou kumukuai Aʻole e oi aku mamua o 75 rubles no pack.

Reviews o ka la hoomalolo

No laila, ma i ka ninauʻano nui. He aha e mea, manaʻo e pili ana i ka lāʻau lapaʻau huahana "Relpaks" nā mea kūʻai mai a me ko lakou mau kumu? He aha nō nā pros a me ka hooluolu mai i keia k? Ka mua mea e olelo ka mea, ma kahi o 80% o nā nā mea i paneʻia - o ka kiʻekiʻe ka hoʻokōʻana o nā huaale "Relpaks" a hiki i loa migraine hoouka. Manaʻo Kōkua mai nā mea maʻi, ma hope o ka lawe wale kekahi Akala a ka eha hele aku ma hope o 30-40 minuke. About 8% o nā mea kūʻai mai anamanaʻo hōʻike ia ma hope o ka hoʻohana 'ana o ka loiloi mua mahele lāʻau o ka 40 mg iʻikeʻia symptoms e like me tremor o na lala, a tingling i loko o ka maka a me ka lima. Eia naʻe, i kēia mau hanana kaʻawaʻawa loa i wahi no, elua no hora ole kekahi hana no hoi ia.

Emi iho malalo o 1% o ka hoʻomanawanui iki mai ka poe i ua ia i ka lāʻau "Relpaks", ka mea mua? Eaia ua i ikeia ma nā mea a pau o kona kanawai. One-kolu o ia ka wā hou-pono o ka lāʻau i i kona kanawai, a me na mea e ae i haʻakoiʻia e loaʻa i ka hope.

Mau loea, e hoailona oukou i waena o ka pono o ka makaukau o kona mehana kanawai ma luna o na moku koko o ke poo. Naʻe, ka mea, e hoailona oukou ia i ke ano o ke ahiahi, i ka loa nīnūnēʻaoʻao 'ole ka hoʻomanawanui e pono e hiamoe. Kēia e e lawa no a pau na kaʻawaʻawa loaʻike manaʻo o ka mea i hala. Mākaukau nō hoʻi i keʻano kēia: ma ka Akä naÿe, e like laau lapaau, i mea ole i kekahi hapa o ka eletriptan lāʻau "Relpaks" nui maʻalahi tolerated migraine kanaka.

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