Ola kino, Hoomakaukau
Ka lāʻau "Sulpiride": hōʻike manaʻo, nāʻikepili, analogs
Psychosis o ka loli iki ana oolea pu manaʻo kanaka a mau loa aku. Over na kenekulia ka mea i manaoio aku i uluhia e ka daimonio i loko o ka maʻi kanaka, a no ia mea, "hoolaia" keia pilikia i Ua kūpono. Prior i ka haku o neuroleptic ka lapaʻauʻia kokua o psychiatric kāna hana he lāʻau lapaʻau'āpana hana e hoʻomohala i ka kumu o belladonna, henbane, opiates. Hana e like me ka hana maikaʻi me ka kalipuna (intravenous) a bapetizoia i ka hoʻomanawanui i loko o ka moe lāʻau.
Ka loa mua antipsychotic chlorpromazine hiki ke kapaia, a i 'Imi ia no ka iapaau ana o nā mea maʻi me ka noʻonoʻo' pilikia mai 1953. Currently, i ka papa inoa o antipsychotic lapaʻauʻia, antipsychotics me ka nui loa hoʻonui. Kekahi o hoʻomano i hoʻohana ai 'o keia pae ka "Sulpiride". E hoike kakau ia e like me ka lahui atypical antipsychotic.
pharmacodynamics o ka lāʻau
Neuroleptic hookoia "sulpiride" antidofaminergicheskim pili i ka hana, m. E. Ma ka Central ko mākou hopohopo'ōnaehana lāʻau ālai 'ʻano nui dopaminergic receptors. Dopamine mea nui i ke keʻena o ka "uku'ōnaehana" o ka lolo - stimulates ka makemake ka waiʻona ma, satisfying ma mua, ma ka huli, e loli ai ka keʻano o ka hanaʻana a me ka hoʻonaʻauao motivational. Ma kiʻekiʻe lawa nā māhele, hua mai la i loko o ke kaʻina hana o kekahi maikaʻi hana (ma ka pilikino manao o kekahi kanaka) -? Eaia o ono ka ai, ka ke keka,ʻaʻoheʻoluʻolu ke kino o ka waiʻona ma ke. Me ua hou i ka ulu nui o dopamine i loko o ka Central ko mākou hopohopo'ōnaehana manaʻoʻike oluolu, a me ka emi - hoʻomōhala symptoms o ke kaumaha.
Hana "sulpiride" ma ka mahele lāʻau e oi 600 mg (i kela la nui o ka lapaʻauʻia) mea he antipsychotic ano. Inā na dosages emi o 600 mg - oi prevalent stimulant a me antidepressant 'ole. Naʻe serotonicheskie, histamine, adrenergic receptors lāʻau, he uuku ia.
Lapaʻauʻia - analogues
Ka medicament "Sulpiride" - atypical neuroleptic, no a hiki i ka pae ana o hookomoia benzamides - i ka pono nui helu o ka lapaʻauʻia i mea like ma ka haku mele 'ana, a mai ka hopena. Aia mau ai 'e like me ka lula ATC 4th pae. Mau mea i ka "Betamax", "tiaprid", "Eglonil". Kaawale mai kēia mau mea, he palahalaha consumer koi "Prosulpin", "Eglek" "Restful" "Vero Sulpiride", "Sulpiride Belupo." Reviews no a pau na laau lapaau ma nā mea kūʻai mai hiki i nā maikaʻi kuhikuhi a me ka io. Ua pau hilinaʻi nui ma luna o ka oolea o ke ahonui o ka moku'āina o ke ola, i kona pā lonoaʻili i ka papa kuhikuhiEʻeleu 'Oponopono - sulpiride, a me ka laʻau heluna o ka lāʻau' ia, e loaa ia ia ke kauka.
Nāʻikepili e loaa ka lapaʻauʻia
Sam neuroleptic "Sulpiride", kona analogs i ke 'ano palahalaha poepoe o ke keiki, a hiki ke häʻawi mai ai iä loaa i ka maʻi i lawa nui. E lawe ia i loko o ke alo o ka schizophrenia i loko o ka huʻi kahua o ka hoʻonaʻauao, a me ka wā e ka maʻi. Sulpiridsoderzhaschih hoomaikai aku la lakou i ka hoʻohana 'ana o antipsychotics i ka huʻi ke kahua o ka hooulu ana o ka delirium (ka noʻonoʻo kāna hana o ke ano, pu ma ka haunaele o ka ike paka i HEN, mai pōniuniu, a hiki coma). Muli o kona kulana pinepine i ka lāʻau 'ua hoakaka ia no kela neurotic kāna hana, a kaumaha, nānā' ole o ko lākou mau kumu.
I ka vertigo o kekahi kumu i ke heluhelu lawe "Sulpiride" manual. Reviews o nā mea maʻi a me ka 'inikua nā limahana e pono wehewehe aku medicament i loko o ka hana maikaʻi i vestibular neuritis, ka wā hoʻokō' ole 'vertebrobasilar-basilar' ano me ka otitis Media, a me cranial traumas, me Meniere ka maʻi (hoonuiia ka leo o ka loli i loko o ka pā pepeiao lua, a waiho puʻe ma na keena kuleana no ka malama ana equilibrium i ke kino a me kona kohoʻia i loko o ka lewa).
E like me ka "Sulpiride" hapa o ka hulina Inc hiki ke hoʻohana 'ia i loko o pākōlea hana no peptic ulcer maʻi a me ka nanaina aku na naau oʻu maʻi pale.
Owai la ka mea e hoomanawanui, mai ka lalau ana antipsychotic ai 'ma ke kumu o ka sulpiride?
Neuroleptics "Sulpiride" lāʻau analogues o ka papa hana 'Oponopono mai i kekahi papa inoa o nā contraindications. Mai lawe ia i kanaka me ka hypersensitivity e sulpiridu, a loaa mai ka hyperprolactinemia (me ka nui loa ke kiekie pae o ka hōmona prolactin i loko o ke koko). Alaila, ua ole ia keia k me ka prolactin-e kaukaʻi hikoko (umauma Ka maʻi 'aʻai, prolactinoma pituitary gland , etc.).
Eia, "Sulpiride" (nāʻikepili i ho'ākāka 'ia ma luna) ua papa aʻo i loko o pheochromocytoma (hormonallyʻeleu chromaffin aeea hikoko), manic psychosis a me kela affective kāna hana me ka' ano 'aggression epilepsy. Mai ka hoʻohana i kēia ka lapaʻauʻia sulpiridsoderzhaschih ku ei ka backdrop o huʻi waiʻona intoxication, kaʻapu kōheoheo me hypnotic lāʻau lapaʻau ai 'a me narcotic analgesics.
'Aʻole e hōʻike' ia o ka hoʻohana 'ana o ka neuroleptic "Sulpiride" e hoomanawanui i elemakule ma lalo makahiki 18 a me na wahine i lactation.
Hikiʻaoʻao waiwai o
Adverse reactions e neuroleptic ia ia iho, a analogues "sulpiride" ahonui e hoike, a ola 'Oihana i emi iho e like me ka lawa nui, me ka nui loa worsening i ke ano o ka hoʻomanawanui iki mai. Aia He He manawa kūpono o ka hyperprolactinemia i loko o ka likeʻole ma o nā 'ano apau loa (gynecomastia, dysmenorrhea, frigidity, hoemiia potency, galactorrhea, mahuahua ma ke kino paona).
E möakäka hou hiki hoike ana o ka extrapyramidal maʻi pale, a ua hoikeia mai ma ka pathological kāna hana o ka nui a me ka pono o ka noho'na makaainana i ulu neʻe hua mai ma skeletal nāʻiʻo, hoʻololi i Muscle leo. Eia naʻe, lōlō mea,ʻaʻole he symptom kēia e hōʻoia ana i ka oiaio o extrapyramidal maʻi pale.
E like me kaʻaoʻao reactions i "Sulpiride" analogs neuroleptic, e hana tremor, akathisia (hikiʻole e ia i maha), dyskinesia, Kanikani'āʻula, drowsiness, uunu nui kiʻekiʻe excitability, irritability. Hiki ke hoike mai symptoms o neuroleptic malignant maʻi pale, wehewehe aku ma autonomic abnormalities, paleʻili, hyperthermia.
ʻaoʻao 'ole, mai ka gastrointestinal'āpana i ia i ka waiʻona ma o dryness i loko o ka waha, no ka hooulu ana o ka heartburn, nausea helehelena, retching, constipation. Hiki ho'ā hope o hepatic transaminases a me kona'ākilikai phosphatase.
Mea'ōnaehana mānowai koko'ōnaehana palapala noi "sulpiride" hiki pane ka hoomahuahua i loko o ke koko, (kākaʻikahi - he emi i loko o ke koko,, pōniuniu), mahuahua naau ana, a mahuahua nui QT-wā mawaena. Loa kākaʻikahi, akā, e hiki lohe ia ma luna o ka "Sulpiride" lāʻau pane mai lapaau hōʻike i ka hooulu ana torsadedepointes 'ano o ka arrhythmia.
Allergic hoike ana e like me ili poʻe noʻonoʻoʻole, pruritus, eczematous lesions. I kekahi manawa oe e lohe e pili ana i ka 'aʻe' ana o pilikia makapō acuity.
dosing a me ka noi aku a puni 'ano paha
E like me na olelo ao no ka hoʻohana ana i ka medicament, nō kāu kanaka makua e hoomanawanui i ke kaumaha ma muli o ka maʻi hoakaka ia mahele lāʻau o 100-300 mg no lā (māheleʻia i loko o nā māhele 2-3). Una pāʻoihana lawelawe i loko o kekahi laʻau heluna: 100-800 mg no lā no intramuscular aaieieno? (Ma mua i pono e lulu). Ke i kā mākou tolerated mahele lāʻau no i kanaka makua, he 1,6 g.
Inā ka mea i pono, e hāʻawi aku "sulpiride" i na keiki ma lalo o makahiki 18 o ka makahiki, i ka laʻau heluna E e pōpilikia e lawe i ka mooolelo o ka kaumaha ma luna o ke kumu o ka 5 mg no kilogram o ke kino ke kaumaha.
Inā i ka hoʻomanawanui i ke ano o ka psychosis i loko o ka huʻi paha maʻi ke kahua, Inc nō kāu hoʻomaka me intramuscular aaieieno? (400-800 mg kela la i keia). Ma ka hapanui o na hihia, i ka wā o ka iapaau ana mea ma ka liʻiliʻi 2 pule. A hiki i ke ola o ka hoomanawanui, ma ka intramuscular ka pahu kui hoololiia a hiki i ka? Eaia "sulpiride" i loko o ka Akala a. Neuroleptic "Sulpiride" hoʻomanawanui hōʻike manaʻo wehewehe me ka mana ka lapaʻauʻia. Duration o ka papa o ka Inc hiki e hooponoponoia ia mea, a me ka hoʻololi wale ma ka hele kauka.
Excessive nā māhele
I kekahi manaʻo symptoms e hoike ana i ka oiaio o ka loa i ka i kā mākou ana nā māhele luna,ʻaʻohe. IeAUPIIe, IAa IO i loko o kēia mau wahi, i hiki, he mea hoʻomāhuahua mau ana i ke koko,, blurred hihio. Paha i ka hooulu ana o ka sedation (suppression o ka ike paka i hoʻonāukiukiʻia ai ', hoʻomālielie i hookoia, oiai kiekie nā māhele - hypnotic). Ma ka hapanui o na hihia, ka ona o ka lāʻau "Sulpiride" ahonui e hoike hōʻike i keʻano o ka nausea, maloo waha, mahuahua sweating, ka luaʻi. Ma pohihihi keia hihia hoʻomōhala extrapyramidal symptoms, gynecomastia hiki i hoʻomaka ai kane hoʻomanawanui iki mai (umauma hoʻonui). Loa kākaʻikahi olelo i haʻi parkinsonism, coma.
Like e wae antidote no "sulpiride" i kahi waiho, symptomatic lapaʻau ua paipaiʻia, ke kaumaha ma muli o ka ano o ka hoʻomanawanui. Ma kekahi mau hihia, pili holinoblokatory kikowaena hana.
Ma mea e hoʻolohe ana i?
Loa nā huahana antipsychotic pūʻulu (me sulpiridsoderzhatsie "Betamax", "Vero Sulpiride", "Prosulpin", "Sulperid Belupo", "Eglonil", "Sulpiride") hōʻike manaʻo hoʻomalu a me nā pae'ōnaehana kuhikuhi, a ua papa i ke kāʻei kua o ka waiʻona nā mea inu. No nā mea maʻi me ka epilepsy ua? Aeiiaiaoaony e hoʻomaka lapaʻau a me ka electrophysiological haʻawina i ua sulpiride emi i ka paepae puka i kāʻili 'ana i hope. Inā ka lāʻau e hoʻohana concomitantly me ka ai 'e hoomahuahua i ka pilikia o ka ventricular arrhythmias, e like me nā mea maʻi pono maʻamau ka mālamaʻana o ka electrocardiogram. Hoomahuahua ae la lakou QT-wā mawaena hilinaʻi nui ma luna o ka mahele lāʻau.
Inā i lapaʻau, "sulpiride" he symptoms o hyperthermia (ka mea e kuhikuhi mai la lakou i ka ulu ana o neuroleptic malignant maʻi pale), ma ka hoʻohana 'ana i ka lāʻau e ke hele.
Koke cessation o Inc "sulpiride" hiki hoʻonāukiuki withdrawal symptoms. Maltitol mea i loaʻa i loko o ka lāʻau i mea hiki ole e hoʻohanaʻia e kanaka e loaa ana mai ka fructose intolerance.
Iloko o ka holoʻokoʻa iapaau ana au e e wary o kaa a me ka manaʻo o ka hooponopono ana e noi ana kokololio muli o psychomotor a me kiʻekiʻe lehulehu.
Sulpiridsoderzhaschie lapaʻauʻia a me ka hāpai keiki
Women i hāpai keiki "Sulpiride 'hōʻike manaʻo i koe i loko o ka loa maikaʻi kuhikuhi. I kā mākou allowable mahele lāʻau no ka hapai wahine, he 200 mg no ka lā i ole hoʻonāukiuki teratogenic 'ole (deflection o embryonic? Acaeoey). Na kŘpa a nui nā māhele o ka lāʻau no ka hapai wahine No 'ike i loaʻa. No hoi, aole hoi heʻikepili ma o ka Loaʻaʻia hopena o ka ai '-antipsychotics ma lolo kūpono' ana o ke keiki.
I mau, ola ka poe makemake ole e hoʻohana "Sulpiride" no ka iapaau ana o ka hapai wahine, koe nae ma ka manawa, kahi i maikaʻi ia no na wahine ka i lanakila ma luna o Loaʻaʻia kamepiula a hiki i ka fetus. Ma ia mau hihia, "Sulpiride" aʻo (hōʻike manaʻo paramedics hookupaa iho la ia) i ke heluhelu lawelawe i loko o ka lalo hiki nā māhele, a ina he mea hiki, e kń i ka wā o ka nohoʻana.
Ma na keiki i hanau i na wahine e lawe i hāpai keiki sulpiridsoderzhaschie lapaʻauʻia kēlā wā i kēia wā malama gastrointestinal symptoms (bloating, a no laila, ma luna o. N.) Associated atropinopodobnye ole o neuroleptics. I kekahi manawa oe e lohe e pili ana i extrapyramidal maʻi pale. Ma breastfeeding hookipa ana "sulpiride" contraindicated.
Manao o nā mea maʻi "sulpiride"
Ke bulk o ka hoʻomanawanuiʻana ma luna o ka lāʻau "Sulpiride" hōʻike manaʻo koe he maikaʻi ao ao. Neuroleptic lawa pono a me ka hoapono aku i ka hai aku ano. People lawe "Sulpiride" a me kona analogues no ka noʻonoʻo 'symptoms iloko o gastric ulcer a duodenal ulcer, hai mai la i ka emi i loko o ka nui o abdominalʻeha a me ka hana hou i loko o ka mau kulana.
Small puke o ka medicament (50 a hiki i 300 mg i ka lā) e pinepine hoakaka i nā mea maʻi e loaa ana ma hoopii o pinepine pōniuniu i kupu mai no kela kumu. Ke bulk o kēia mau hoʻomanawanui iki mai ua māʻona i ka hopena o ka lapaau.
Nui nā māhele "sulpiride" (oi ma mua o 600 mg no ka lā), ma ka manao o ka 'inikua poe hana i ka hoʻolako' ana i ka hoʻokō antipsychotic hopena ma luna o nā mea maʻi. Nā māhele emi o 600 mg, a ma ka manao o ka lapaau a me nā mea maʻi, lawe noho haumāna kahi a me ka antidepressant hopena.
Aia o kekahi pūʻulu o nā mea maʻi i haʻalele i ka "sulpiride" i loko o ka io ala. Mai kanaka hoʻomōhala nausea, pīhoihoi, giddiness. Noke symptoms nalowale ma hope o discontinuation o ka "sulpiride".
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