Ola kino, Hoomakaukau
Na Ke Kumu no ka hoʻohana "tiapridal". Analogs a me nā hōʻike manaʻo
"Tiapridal" - antipsychotic ka lapaʻauʻia ua hanaʻia ma ka tiapride. Ka lāʻau 'Ua noi me he kiaha dala, analgesic a me hypnotic. Kumu o antipsychotic hana - ka paleʻana i ka dopamine receptors, a me ka nui loa pili i ka functioning o ka CNS. Ma keia 'atikala, ua wehewehe mai i loko o au mamuli e pili ana i ka waiʻona.
Haku mele 'ana ec i ka lāʻau
Ke lapaau mea i loaʻa i loko o nā 'ano apau loa, ke papa hiki ke kuai, a me ka pāʻoihana.
- Kekahi papa me kekahi ampoule maupaʻa 100 milligrams o ka papa kuhikuhiE ke keʻena a me kākoʻo 'ona. Like kākoʻo nā mea hoʻohui hoʻohana ma o ka haku mele 'ana o ka povidone, makanekiuma stearate, mannitol. Ka haku mele 'ana Ua pū inā me ka koʻana koko colloidal'okikene lua, silikone a me ka microcrystalline kelulose.
- Kaawale mai na kumu nui ke keʻena o ka pāʻoihana maupaʻa paʻakai koloriside a me ka wai no ka pahu kui.
I kekahi pahu, he 20 na papa (2 blisters me 10 o na papa io) a 12 hue (2 blisters o 6 hue). Na Ke Kumu no ka hoʻohana "Tiapridal" i loko o ka palapala o ka pāʻoihana no ka pahu kui E ho oku ui lawelawe intravenously a intramuscularly. Kēia palapala no ka lāʻau mea pono wale no o ka iapaau ana o kanaka makua nā mea maʻi.
Pharmacodynamics "tiapridal"
Ke medicament i neuroleptic, analgesic a me anxiolytic hana. E like me ka manual, "Tiapridal" selectively ālai 'ka functioning o D 2 receptors o kikowaena dopamine. Pela ma D 1 receptorsʻaʻohe like me ia. Ka lāʻau 'ʻia pakele o ka psoriasis, ka wā hoʻohana' ia ma o nā kūpuna? Ienoai aa noʻonoʻo.
Pharmacokinetics "tiapridal"
ua ia akulla Intramuscular hooponopono o ka lāʻau (200 mg) o kona i kā mākou piʻi i loko o ke kino ma hope o 30 minuke, ka hoʻohana 'ana i ka papa ma ka ia mahele lāʻau - 60 minuke. Ke bioavailability o ka lāʻau ka wā hoʻohana koke me ka 75% muaʻai mahuahua i 95%. No ka mea, ai 'ia ana, piʻi pū a me kona i kā mākou piʻi i loko o ka meaola (40%).
Omo i loko o ke kino o ke kua'āina o ka poʻeʻelemākule nā mea maʻi. "Tiapridal" kauoha no ka hoʻohana pili i ka Agena nā keʻa i ke placental a me ke koko-lolo o ke'ākeʻakeʻa mai. Ua ua ike ia i ka iapaau ana i ka lāʻau 'mea i loaʻa i loko o ka haku mele' ana o ka umauma o ka waiu. Ma nā wāhine, ka hapa ana o ka lāʻau wikiwiki ma mua ia o na kanaka (ma 2,9 hola), ka like o 0,7 hola. Pūnao wehewehe aku me lōpū. Ke kumu nui loa o ka lāʻau (70%) ua wehe 'ia mai ke kino ma na puʻupaʻa ua hoʻololiʻia.
Nāʻikepili "Tiapridal" hoomalolo
E hoʻokō i ka Inc me ka ai ' "Tiapridal" heluhelu like penei:
- dyskinesia (tardive, noho'na makaainana i ulu);
- Gilles ka'Aroda: Tourette maʻi pale;
- chorea;
- 'ano' kāna hana (ʻano pākīkē moku'āina, manaʻo pīhoihoi listen AL.), kūpono ma ka paa pele o ka maʻi alcoholism a me ka poʻeʻelemākule nā mea maʻi;
- hopena maikaʻi 'hoike ana ma ka hana, e like meʻano pākīkē moku'āina a me ka manaʻo pīhoihoi;
- eha mālama nui ano (maʻi ano).
Contraindications, hoʻokau 'e loaa "Tiapridal" lāʻau
Ua papa i ke kau ana o "Tiapridal" kauoha no ka hoʻohana no ka poe mamo nona ka makahiki ka emi o na makahiki eono. Ma pediatric Inc ua lawe mai wale Akala. Ka lāʻau 'E ole e hana wale aku nā wāhine a me nā mea maʻi i e breastfeeding. ua i hoʻohana 'ia ka lapaʻauʻia ma ka hihia o ka hypersensitivity i kona eiiiiiaiou, a me kekahi mau mea. Contraindications nā mea Hawaii:
- hepatic a me kaʻaʻa puʻuwai 'ole, a he nui ka oolea;
- prolaktinzavisimogo diagnosing hikoko, e hoʻohuoiʻia o kona alo;
- hypertensive hoʻoponopono ulia;
- ʻike, o ka pheochromocytoma, he hoʻohuoiʻia no kona ola.
Papa a me ka pāʻoihana ua hoʻohana pū me "sultopride" a me ka dopamine mea loaʻa agonists (i ke koe o ka iapaau ana o nā mea maʻi me Parkinson ka maʻi) ka mea, i hui ia me kekahi mauʻano o nā neuroleptics, Anati-arrhythmic Luna o ka papa au, a III A.
Medicating "Tiapridal" ke aʻo 'Aʻole i' ae ka poʻe hoʻohana "Moxifloxacin", "sparfloxacin", "Difemanila", "Erythromycin", "bepridil," "mizolastine", "levodopa", "cisapride" a me ka intravenous "vincamine" .
Inā ka hoʻomanawanui (oi loa ka kūpuna) ua malamaia lakou nei, me ka ai 'i e alakai ai i ka hooulu ana o ka hypokalemia, cardiac conduction mea hōʻemi, hooloihiia mai QT wā mawaena, ka hanana o bradycardia i olelo ia ano, e hoʻohana i ka "Tiapridal" pono e akahele. Mālama nui ua koi ia ma ia hihia.
- Parkinson ka maʻi;
- congenital QT wā mawaena elongation ano;
- hypokalemia;
- maʻiʻaʻa puʻuwai ole;
- bradycardia;
- maʻi i loko o ka mea o Nyos i ka mea'ōnaehana mānowai koko'ōnaehana (decompensation anu u);
- epilepsy.
Iapaau ana me "Tiapridal"
ma ka noi o "Tiapridal" e manual i ke heluhelu ka hoʻohana 'ana i ka mua ma ka liʻiliʻi nā māhele, ke kiʻekiʻe o mahuahua ia lakou, i mea e loaa i ka i kā mākou hopena.
'ano' kāna hana
No ko lakou kokua mea pono e pili 200 mg o ka lāʻau i kela la (mai ka 300). Ka mea maikaʻi hookoia ua loaʻa i loko o eono pule ma luna o kaʻawelike. Mua e hoomanawanui i lawelawe i ka haʻahaʻa mahele lāʻau o ka lapaʻauʻia - 50 mg. A hookahi mahele lāʻau E e hoʻopau palua i ka lā, a me kona mea ulu ua aeia'ku ia ma kaʻaeʻana me ka ke koho 'ia wā mawaena, o ka hana ua hana ke kiʻekiʻe, e lawe i ka mooolelo akamai'ōlelo aʻo. Na kela la i keia mahele lāʻau E ole mamua o 300 mg.
Maʻi, pili ka eha
Na kela la i keia mahele lāʻau o ka lāʻau no ka iapaau ana o ia mau rula mea mai ka 200 a hiki i 400 mg.
Chorea, Gilles ka'Aroda: Tourette maʻi pale
I ka lawe ana mai i ka iapaau ana o ke keiki i kela la mahele lāʻau ua koho e lawe i ka mooolelo o ka kino kaumaha, a ma kahi o 3-6 mg / kg. Inā 'oe Pono e hoʻomaka i ka makua Inc, mua hoʻohana 25 mg o ka lāʻau no ka lā, ma hope (ma hope o ka gradual mahuahua ma ka mahele lāʻau) - 300-800 mg.
Manaʻo pīhoihoi, aggression
Ke paipai kela la i keia mahele lāʻau o ka medicament mea mai ka 100 a hiki i 150 mg.
'ano' kāna hana
Ke paipai mahele lāʻau no ka ao, i (mai ka 200 a hiki i 300 mg) i loko o ka hihia o delirious Hawaii paha predelirioznogo e pii ai a hiki i 400-1200 mg. ʻO kā mākou hiki mahele lāʻau i pono ole e oi, o 1800 mg. I ka hoike ana o ka lāʻau hua ma luna o kaʻawelike hola kela elima. Inā iapaau ana mea e pono ai ka mea kūpuna kanaka, i kela la i mea 2-3 injections ma waena o i malama wā mawaena o 6 hola. No ka iapaau ana o ia nā mea maʻi paipai kela la i keiaʻai ana o ka 200 a hiki i 300 mg o medicament i kekahi manawa ua 'ae' ia e komo i emi ma mua o 100 mg "tiapridal".
, Pili olelo o ka maʻi 'ano o ka eha
Therapies ka nānā 'ana ma luna o ka lawelaweia ana o kela la i keia mahele lāʻau e like me 200-400 mg o ka lāʻau.
ʻaoʻao 'ole ka wā lawe "Tiapridal" lāʻau
I ka hana maikaʻi lāʻau "Tiapridal" manual, hōʻike manaʻo hoʻokūpaʻa i ka likelihood o kekahi adverse reactions. 'Aʻe' kānāwai i loko o ka urogenital, ko mākou hopohopo, endocrine a me ka mea'ōnaehana mānowai koko nenoai. Eia hou, aia no he pilikia o ka pilikia a me ka makaukau. No nā hopena maikaʻi 'ole nā allergies, ili hoikeana pu ma ke kaupaonaʻana, ka waiwai, orthostatic hypotension.
Overdose "tiapridal"
Inā 'oe hoʻohana excessive mahele lāʻau hiki overdose a me kona symptoms nā haunaele o ka ike paka i, ka loa kaumaha o ka a - coma, neuroleptic maʻi pale (malignant, huʻi pepa). I mea e hemahema i kēia moku'āina o ka meaola ua lawe mai iapaau ana me ka nānā 'ana ma anticholinergic konohiki. Ma hope iho o ka abolition o ka lāʻau e pono e lawe mai symptomatic lapaau a me ka plasmapheresis.
Cautions
Mua i ka lapaau "Tiapridal" manual ia kekahi e paʻipaʻi hypokalemia. Ma Inc ia mea nui ia mau kanaka hoʻoponopono electrolyte kaulike, hoʻomaka ka electrocardiogram, kanaka hoʻoponopono i ka lapaʻau kiʻi hou.
Inā he mea pono e pili anticholinergic ai 'ka hopena e loaa ana neuroleptics extrapyramidal maʻi pale ulu kahi o ka dopamine mea loaʻa agonist.
I ka manawa o ka iapaau ana e haʻalele hana e ho oweliweli kekahi ikehu hoʻoweliweli, ka mea, ua i paipai i ka hana hana e noi ana kūikawā a me ka poe ola, pane.
AaOIeIOUIeXAOAaIN a me nā waiwai
Kekahi hui malu pu ana hoʻomākaukau me ka lalau ana ka lapaʻauʻia "Tiapridal" ke aʻoʻia, manaʻo pili i ka pahiki o ka hanana o undesired reactions. Ua UaʻAʻole pono i lapaʻau noi "Clonidine", antihistamines, anxiolytics, barbiturates a me opioids, like "tiapridal" kanawai e e hou hai. Manawa i ka incompatibility E ole e lawe "levodopa" a me ka waiʻona. Ka lapaʻauʻia hiki ke hui me ka hoʻohana 'ana o neurotrophic ai', analgesics, antidepressants, neuroleptics. High kamepiula o orthostatic hypotension, he mea ka i ka wā hoʻokahi pono o antihypertensive ai 'me "Tiapridalom".
Ke kāki o ka lāʻau analogues, hōʻike manaʻo e pili ana i ka lāʻau "Tiapridal"
Inā pono lapaʻau "Tiapridal" 'o ia hoʻi ke aʻo hōʻikeʻano e oe i mea i ka lāʻau o. Ke kumu kuai o ka ai 'o ka nui i loko o ke koho ana o ka medicament no ka lapaau. Ke kākoʻo pāʻoihana ma na hue hiki ke kūʻai no ma kahi o 995 rubles, a me nā papa - no 1.400 rubles.
Mawaena o na analogues o ka lāʻau - "Eglonil", "Betamax". O na pani ai i ke koho "Sulpiride" a me "Prosulpin". Aia i kekahi mea like o ka lāʻau - "tiaprid", oia ua noʻonoʻo i ka loa ho'āmana, ia mea hala loa he kaulana koho, na wahi lulu lāʻau? Iecaianoaaiiie i epa me ka poe "aloha". E like me ka hapa o ka "tiaprid" haawi i ka iaʻeleu waiwai, i ka hapa o ka lapaʻauʻia "Tiapridal". 'Āpana analogs kuhikuhi ia kekahi e koho, i ka wa a ka mua hiki ole e hoʻohana ka poʻe me kekahi ai 'ke kumuʻaoʻao' ole, a 'aʻole i kekahi i makemake ai. I ka lāʻau 'ua loa ka hoʻokō, lawe i mooolelo nui o na kumu i ka wā i koho.
Ma lapaʻau, ia mea nui, e hahai i ke kauka i ka'ōlelo aʻo, a koi, a ÷ kuhi no ka hoʻohana. "Tiapridal", e like me ka hoike ma ka manaʻo, ma ka hapanui o na hihia, ua hoʻohana 'ia e hoʻopau i ka olelo pu ma ko mākou hopohopo pīhoihoi, aʻano pākīkē hana, kanakaʻona mau psychosis. IeAUPIIe, IAa IO, nā mea maʻi a me na kumu e maona i ka hopena o ka Inc. Holo nōhie, he refresher papa ua i koi 'ia no ka mea, i ka makemake kanawai ua ulu ma hope o ka hoʻokō' ana o ka papa mua. Reviews hōʻike i no nā mea maʻi lapaau "Tiapridal" oluolu e hoʻohana.
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