Ola kinoHoomakaukau

Antidepressant "Velaksin": ahonui e hoike, aʻo no ka hoʻohana 'ana, analogs

Hiki au e kuai antidepressants me ke kuhikuhi? A papa inoa o ia huahana mea,ʻaʻole nui. O ke kumu ho i ka mea i ka mea, hiki e addictive, a me ka poʻe koa o kaʻaoʻao loa. No laila, ma mua ka lawe ia mau mea, eʻoiaʻiʻo, e kipa i ka hoʻomalu.

kekahi mau 'ike

Kaumaha ua iʻia ma ka ai '. Akā, e hoʻoikaika i ka functioning o ka'emi oihana, he nui na kauka nō i koi 'ana i kā lākou nā mea maʻi likeʻole antidepressants. Kekahi o ia mea i ka lāʻau "Velaksin". Hoike e pili ana i keia mea paahana a me kona hiʻona a me nā'ōlelo aʻo no ka hoʻohana 'ana, e e hōʻike mai iā ia ma lalo nei.

I ka haku mele 'ana o ka lāʻau, kona ano o ka? Iecaianoaaiiuo

Ma ka palapala ia produces he antidepressant like "Velaksin"? Papa a me nā capsules - i nāʻano wale o ka lāʻau.

Papa "Velaksin" i keʻokeʻo, kahakahaia ma kekahiʻaoʻao "E741", a me ka hoʻopoepoe i lalo shape a me ka chamfer. Kā lākou hana 'Oponopono ka venlafaxine, i ua poe ma ke ano o ka hydrochloride. I hookomoia ma keia ka lapaʻauʻia nā kākoʻo eiiiiiaiou e like me colloidal ka silica i anhydrous, lactose monohydrate, paʻakai pia glycolate, makanekiuma stearate a me MCC.

Piha o na papa io o blister he huihui 'a me cartons pakahi.

Uluwehi O "Velaksin" - capsules, olelo ao no ka hana i mea e hoʻopuni ana i ka'ōpala, pepa, gelatin a me ka paa. Ka mea, i 'alani-eleele chap, a me ka colorless kūpapakū. Kaʻeleu ke keʻena o keia palapala Ua hoi he hui venlafaxine. Ma waho aʻeo ia i kona haku mele 'ana o kēia ka lapaʻauʻia nā aiiieieoaeuiuo iiauo nā mea hoʻohui.

E like me ka lāʻau hana?

"Velaksin" - he hou hanauna o Anati-depressant. E like me ka Nine Inch 'ole o konaʻeleu waiwai, aole ia i hui ole ia me kekahi ike papa o antidepressants (e laʻa me, tricyclic, tetracyclic, a me' ē aʻe). Kilo'ōlelo aku nei au i ka lāʻau meaʻeleu enantiomer 2 racemate.

I ka rula o ka hana ana o keia k ua pili i kona waiwai, e potentiate i ka CNS nā aʻalolo impulse EYI.

E like me na kuhikuhi, venlafaxine a me kona nui metabolite (EFA ole O-desmetilvenlafaksin) ho i potent nā mea kūpale o ka reuptake o norepinephrine a me ka serotonin a me ka nawaliwali nā mea kūpale o dopamine reuptake. Mākou hiki ole ke olelo i ka mea hiki ke emi i ka Hoʻokolohua-adrenergic ha awina ma hope o ka hookahi, a ikaika aku ka lapaʻauʻia i kēia mau waiwai. EFA a venlafaxine e like mana e ku e ia reuptake o neurotransmitters.

He aha hou aʻe mea kupaianaha lāʻau "Velaksin"? Alakaʻi ai ia mau moʻolelo i ka hana 'Oponopono o ka lāʻau i kaʻo Solomona me ka n- a me ka m-cholinergic receptors, lolo α1-adrenoceptors a me histamine H1-receptors. Eia kekahi, e inhibits ka hana o Mao, a maiʻaʻohe similarity me fentsiklidinovymi, opioid, benzodiazepine a me ka NMDA-receptors.

Nā kinetics o ka lāʻau

ina paha i ka lāʻau o ke kemu, "Velaksin" (papa)? Na Ke Kumu no ka ho ohana i hākālia nō i kaʻeleu ke keʻena o keia k ua hala loa pono ke kemu, mai ka gut. Ma hope o ka hookahi mahele lāʻau o ka medicament i loko o ka laʻau heluna o 25-150 mg o kona kiekie lehulehu i loko o ke koko ua hiki aku ma hope o 2.4 hola. Pela venlafaxine ua nui metabolized i ke alahele mua ma ke akepaʻa. Inā ua laweʻia ka lāʻau a me ka ai, oiai kona piko lehulehu, piʻi pū ma 27-30 minuke ma ka wai koko.

I ka papa kuhikuhiE metabolite Ua noʻonoʻo pono i ka mea o ka O-desmetilvenlafaksin. Kona hapa-ke ola a me ka hoʻopau hapa-ola o ka venlafaxine o 11 a me 5 hola, niioaaonoaaiii (ia auoiaea i loko o ua hoʻololiʻia ano ma nā puʻupaʻa).

Nā kinetics o ka ai 'ma kūikawā lapaʻau wahi, i hiki

Uluwehi O "Velaksin" aʻo ua koi heluhelu i loko o kanaka me cirrhosis o ke akepaʻa loaʻa'ē aʻe kinetic hiʻona. koko lehulehu o ka lāʻau, a mahuahua nui i loko o kēia mau nā mea maʻi, a me kona uku o ka excretion, ma ka mea ku ole, hoemiia.

I loaʻaʻa puʻuwai insufficiency,ʻaʻa puʻuwai ka hoʻokō 'ole a me ka lōpū huinaʻae ua hoemi EFA a me venlafaxine, a ua hooloihiia i ka hoʻopau hapa-ola manawa.

Ua E hoi e hoʻomaopopo i ka hoohanau a me ka makahiki o ka hoʻomanawanui, aole ia e pili i ka pharmacokinetics o ka lāʻau ma lalo o noonoo.

nāʻikepili no ka

No ke aha la e ua pono i ka mea paahana e like me "Velaksin"? I ka hana o keia k hōʻike i loko o ke kaumaha o nā kumu (no ka lapaau a me ka prophylaxis).

Bans ka manawa

Ma lalo o ka hiki ole rula hoʻohana i ka lāʻau "Velaksin"? Reviews o nā mea maʻi a me na kumu koi i keia k ua contraindicated e loaa:

  • oiai ka loaa ana Mao nā mea kūpale ;
  • i loa hakuʻala kāna hana;
  • ma ka mahuʻi mua ai hookupaa hāpai keiki;
  • i loa kāna hana o ke ake;
  • i breastfeeding;
  • ma ka adolescence a me ka noho 'ana kamaliʻi, i ka mea, a hiki i ka makahiki o ka nui;
  • me ka kiʻekiʻe pā lonoaʻili i ka waiʻona.

Eia kekahi, e pono ia ia k ‰ i lolelua ka angina, myocardial infarction (me ka lānai hou E neʻe i), hypertension, convulsions mōʻaukala, tachycardia, ke kaupaonaʻana poho, a mahuahua nui intraocular puʻe, huina-panina glaucoma, predisposition e kahe ana ke koko mai mucous, a ʻili, manic Hawaii.

Uluwehi O "Velaksin" (papa): kauoha no ka hoʻohana

Antidepressant "Velaksin" E wale nō e lawe i ka meaʻai. Ke paipai ho mahele lāʻau o ka lāʻau, he 75 mg, i puunaue i ka 2 māheleʻia nā māhele (a laila, 37,5 mg palua i ka lā), i kela lā.

Inā ma hope o kekahi mau pule o Inc, ke hoʻomanawanui i ka ke ano i ole holomua, ua mahuahua no ka 150 mg ka kela la i keia mahele lāʻau i ka lā, i loko o nā māheleʻia nā māhele (a laila, 75 mg palua i ka lā).

Inā ka hoʻomanawanui koi i ka mahele lāʻau kiʻekiʻe o ka antidepressant (e laʻa me, nui depressive kāna hana, a me ka rula e noi ana Inc wahi), a laila, i ka technician hiki i hoʻokohu 'ia 150 mg o ka lāʻau i loko o 2 hola, a laila, ke kiʻekiʻe o hoonui i ka mahele lāʻau ma ka 75 mg (2-3 lā hope) e kū ai i ka makemake hopena.

E like me na kuhikuhi, ka mea i kā mākou laʻau heluna "Velaksina" He 375 mg no ka lā. Ma hope o ka hoʻokō 'ana i ka makemake keia, ka mea hiki ke kiʻekiʻe o kuʻu iho ai i ka palena iki kiʻekiʻe.

Relapse Kāohiʻana a me ka mālama 'ana i Inc

Kākoʻoi ka malama ana o na dala e lawe mai i nā malamaʻeono. Ma keia hihia, no ka lapaʻauʻia ia i loko o ka palena haʻahaʻa nā māhele.

I ka mehanaʻaʻa puʻuwai insufficiency? Iaea dosing regimen ua koi 'ia. Ma ka like maʻi lōpū mahele lāʻau e waiho haʻahaʻa ma 25-50%. Ua E hoi e kaulana i venlafaxine e ole e ia i loko o loaʻaʻa puʻuwai insufficiency, mai 'aʻohe' ikepili ma luna o ka maluhia o ia Inc i ka lā,ʻaʻohe.

Kanaka, ka poe i ma hemodialysis, e loaa 50% o ka mau i kela la laʻau heluna o ka lāʻau ma hope o ka Ahaolelo welau.

No ka mehana hepatic insufficiency? Iaea dosing regimen ua hoi i koi 'ia. I ka wā o ka maʻi mea e e hoemi ma ka 50% lōpū mahele lāʻau. Me ka pili ana i ka loa hepatic ole, ma keia hihia i ka hoʻohana 'ana o ka venlafaxine ua hookapuia.

Ma ka kūpuna, ka lāʻau "Velaksin" E e hoʻohana me ka lōʻihi mālama nui. O ke kumu ho i ka hiki 'aʻe o nā puʻupaʻa. ʻO nā mea maʻi Pono e koi 'ia i ka lalo ka hoʻokō mahele lāʻau. Ma keia hihia, ke hoʻomanawanui e ia ma lalo ikaika 'inikua hooponopono.

Hawaiian antidepressant

Ma ka pau 'ana o ka loaa ana i ka lāʻau' E e manaoia e emi i ka mahele lāʻau i nā (i loko o ka pule). Ua Ua koi 'ia e malama i ke kanawai o ka hoomanawanui, ma ka mea e loa kń i ka pilikia o adverse reactions pili me ka abolition o ka lāʻau.

Ka manawa koi 'ia no ka piha cessation o ka lapaʻauʻia, hilinaʻi nui ma ka laʻau heluna, lōʻihi like' ole o ka Inc a me ka kanaka i kanaka.

ʻaoʻao waiwai

He aha e hiki i "Velaksin" ka hua'ōlelo i makemake 'ole o ka waiʻona? E hoike aku nei au i ka ulu ana o ka poe 'ole' ē aʻe adverse hanana hahai ana i ka hana ana i keia mea paahana hilinaʻi nui ma luna o ka mahele lāʻau loaa.

Ka loa pinepine reactions hoike io ano loaʻa nā kēia:

  • hypertension, ua hoʻemi ikaika loa ka makemake,'āno'ē nā moeʻuhane, constipation, Kanikani'āʻula, nausea, flushing o kaʻili, tremors, ka luaʻi, Muscle cramps, maloo waha;
  • hallucinations, hepatitis, ke kaupaonaʻana poho, tachycardia, hyponatremia, apathy, postural hypotension, pōniuniu, manic naoh, ko mākou hopohopo excitability,ʻale, paresthesia, neuroleptic maʻi pale, nanea ana, serotonergic maʻi pale;
  • mahuahua Muscle leo, ke kāʻili 'ana, dysuria, photosensitivity, urinary ka mālama, anorgasmia;
  • kahe ana ke koko i loko o kaʻili,'āno'ē ejaculation, menorrhagia, ua hoʻemi libido, sweating;
  • thrombocytopenia, noho haunaele, erythema multiforme, mydriasis, Stevens - Johnson, pilikia makapō haunaele, hoʻopōʻino hoao, prolongation o kahe ana ke koko manawa, nawaliwali, ili poʻe noʻonoʻoʻole, luhi, anaphylactic reactions.

Ua E hoi e kaulana ia ma hope o ka abrupt withdrawal o ka noʻonoʻo kaa a ho'ēmi i kona laʻau heluna e hiki i kaʻaoʻao reactions me ko mākou hopohopo irritability, luhi, diarrhea, drowsiness, restlessness, headache, paraesthesias, nausea, hypomania, ka luaʻi, sweating, anorexia, Kanikani'āʻula, maloo waha, uunu nui, a me ka pōniuniu disorientation. Nō kāu, i kēia mau symptoms i mehana, a hele aku me kekahi lapaau.

koi

Kuai ina antidepressants me ke kuhikuhi? A papa inoa o kēia mau laau lapaau mea ole loa nui ( "Prozac", "Paxil", "Despres", "Azafen", "Persian", "amitriptyline"), a me ka lāʻau "Velaksin" ua i komo i loko o laila. E kuai oe ia mea i loko o keʻena kūʻai lāʻau lapaʻau, e hiki wale ma ka Kauka ka kuhikuhi.

Ma mua o ka lawe i kēia ka lapaʻauʻia ma lalo o ka nāʻanaʻana, o ka oi aku nā mea maʻi me ka depressive kāna hana, e noʻonoʻo ke kiʻekiʻe pahiki o suicidal ho'āʻo. Ma keia manao, i ka hoʻomaka o ka lāʻau Inc paipai no ka hoʻohana 'ana i ka palena iki mahele lāʻau, a ma lalo o kokoke loa' inikua hooponopono.

People me ka naʻau i loko kāna hana i lapaʻau me antidepressants e hoʻomōhala manic a hypomanic moku'āina.

Nā mea maʻi e eʻoiaʻiʻo, e ao aku ia oukou i ka mea e koke ike i kekahi kauka ma ka hihia o ka urticaria hehee wale, rashes a allergic reactions hemahema.

Kekahi nā mea maʻi i loko o ka kaʻina hana o ka loaa ana venlafaxine malama i kekahi mahele lāʻau-e kaukaʻi mahuahua ana i loko o ke koko,.

ʻelemākule e hoʻomanawanui iki mai e ke ao o ka hiki 'aʻe' ana i ke ano o ke kaulike a me ka pōniuniu? Acaeoey.

Ma lapaau ana o na dala e pakele lawe kanakaʻona mau kea.

Antidepressant "Velaksin": ahonui e hoike, huahana analogues

He aha kanaka i ka i ana e pili ana i keia k i ke ahonui? Ua nui nā mea kūʻai mai i hoike i ka nui helu o kaʻaoʻao 'ole e hana oiai e lawe i kēia ka lapaʻauʻia. Loa pinepine keia k ke kumu adverse reactions e like me drowsiness, nawaliwali, Kanikani'āʻula, ke kāʻili 'ana,'āno'ē noʻonoʻoloi, kaumaha a me ka hilahila. Eia hou kekahi, kekahi e hoomanawanui i koi ae i ua mau waiwai i koe ma hope o ka pauʻana o ka nohoʻana. No hoi, he nui na mea hoʻohana ohumu e pili ana i keʻano o ka withdrawal symptoms a me kaukaʻi.

He aha e puku antidepressant e like me "Velaksin"? Analogs o keia k uaʻaʻole ia e loaʻa i loko o nā mea a pau drugstores. E like me ka rula, mākaukau mau loaʻa nā kēia: "Venlafaxine Sandoz", "Efevelon", "Alvent", "Nyuvelong", "Velafaks", "Dapfiks", "Voksemel", "Venlaksor", "Vensuert", "venlafaxine".

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